eletriptan (Relpax)

Pharmacokinetics

• may have faster onset than sumatriptan
• metabolized by cyt P450 3A4

Drug interactions

• cyt P450 3A4 inhibitors increase eletriptan
  • clarithromycin (Biaxin), ketoconazole (Nizoral), itraconazole (Sporonox), nefazodone (Serzone), ritonavir (Norvir), nelfinavir (Viracept)

• drug interaction(s) of triptans with SNRIs
• drug interaction(s) of triptans with SSRIs
• drug interaction(s) of methylene blue with serotonin agonists
• drug interaction(s) of linezolid with serotonin agonists

More general terms

• serotonin agonist (5-HT receptor agonist, triptan)

Database

• PubChem: http://pubchem.ncbi.nlm.nih.gov/summary/summary.cgi?cid=77993
• PubChem: http://pubchem.ncbi.nlm.nih.gov/summary/summary.cgi?cid=156849
• PubChem: http://pubchem.ncbi.nlm.nih.gov/summary/summary.cgi?cid=656631